Pharmaceutical Intermediates


 

Sr.No. API APPLICATION INTERMEDIATE OFFERED* CAS NO

1

APIXABAN
1-(4-IODO-PHENYL)-PIPERIDIN-2-ONE 385425-15-0
1-(4-BROMO-PHENYL)-PIPERIDIN-2-ONE 27471-43-8
1-( 4-NITRO-PHENYL)-PIPERIDIN-2-ONE 38560-30-4
ETHYL CHLORO[(4-METHOXYPHENYL)HYDRAZONO]ACETATE

27143-07-3/473927-63-8

2-PIPERIDONE 675-20-7
3-CHLORO-5,6-DIHYDRO-1-(4-NITROPHENYL)-2(1H)-PYRIDINONE 536760-29-9
3-MORPHOLIN-4-YL-1-(4-NITROPHENYL)-5,6-DIHYDROPYRIDIN-2(1H)-ONE 503615-03-0
ETHYL 1-(4-METHOXYPHENYL)-6-(4-NITROPHENYL)-7-OXO-4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[3,4-C]PYRIDINE-3-CARBOXYLATE 536759-91-8
1-(4-IODOPHENYL)-3-MORPHOLINE-4-YL-5,6DIHYDROPYRIDINE-2 ONE 473927-69-4
ETHYL- 1-(4-METHOXYPHENYL)-7-OXO-6-[4-(2-OXOPIPERIDIN-1-YL)PHENYL]-4,5-DIHYDROPYRAZOLO[5,4-C]PYRIDINE-3-CARBOXYLATE 503614-91-3
3-MORPHOLINO-1-[4-(2-OXOPIPERIDIN-1-YL)PHENYL]-5,6-DIHYDROPYRIDIN-2(1H)-ONE 545445-44-1
1(4-AMINOPHENYL)-3-MORPHOLIN-4YL-5,6 DIHYDROPYRIDINE-2(1H)-ONE 1267610-26-3
ETHYL 1-(4-METHOXYPHENYL)-6-(4-IODOPHENYL)-7-OXO-4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[3,4-C]PYRIDINE-3-CARBOXYLATE 473927-64-9
2 APREMILAST 3-NITRO PHTHALIC ACID 603-11-2
3-AMINO PHTHALIC ACID 5434-20-8
3-ETHOXY-4-METHOXY BENZALDEHYDE 1131-52-8
3-ETHOXY-4-METHOXY BENZONITRILE 60758-86-3
3-ACETAMIDO PHTHALIC ANHYDRIDE 6296-53-3
3 ACOTIAMIDE N,N-DIISOPROPYLETHYLENE DIAMINE 121-05-1
4 ARIPIPRAZOLE 1-(2,3-DICHLORO PHENYL) PIPERAZINE HCl 119532-26-2
5 ALOGLIPTIN 2-(BROMOMETHYL)BENZONITRILE 22115-41-9
6 ANCRIVIROC 1-BOC-4-PIPERIDONE 79099-07-3
7 BREXPIPRAZOLE 7-HYDROXYQUINOLIN-2(1H)-ONE 70500-72-0
N-(CINNAMOYL)-3-METHOXYANILINE 127033-74-3
4-CHLORO-1-BENZOTHIOPHENE-2-CARBOXILIC ACID 23967-57-9
4-CHLORO-1-BENZOTHIOPHENE 66490-33-3
1-(1-BENZOTHIOPHEN-4-YL)PIPERAZINE HCl 913614-18-3
8 BUTORPHANOL CYCLOBUTANE CARBOXYLIC ACID 3721-95-7
9 CILOSTAZOL 6-HYDROXYL-3,4-DIHYDRO-2(1H)-QUINOLINONE 54197-66-9
10 CABOZANTINIB 6,7-DIMETHOXYQUINOLIN-4-OL 13425-93-9
4-CHLORO-6,7-DIMETHOXYQUINOLINE 35654-56-9
CYCLOPROPANE-1,1-DICARBOXYLIC DIETHYL ESTER 598-10-7
4-[(6,7-DIMETHOXYQUINOLIN-4-YL)OXY]ANILINE] ACID 190728-24-6
11 CARBOPLATIN 1,1-CYCLOBUTANE DICARBOXYLICACID 5445-51-2
12 CELECOXIB 4-HYDRAZINOBENZENESULFONAMIDE 27918-19-0
13 CRIZOTINIB 4-IODO PYRAZOLE 3469-69-0
14 CARFILZOMIB MORPHOLINE ACETIC ACID HCl 3235-69-6
15 CIZOLIRTIN 1-METHYL-1H-PYRAZOLE 930-36-9
16 DOLUTEGRAVIR/ IMATINIB AMINOACETALDEHYDE DIMETHYL ACETAL 22483-09-6
N,N-DIMETHYL FORMAMIDE DIMETHYL ACETAL 4637-24-5
17 DABIGATRAN 4-(METHYLAMINO)-3-NITROBENZOIC ACID 41263-74-5
ETHYL -3- (PYRIDINE-2YL AMINO ) PROPANOATE 103041-38-9
ETHYL 3-[{3-AMINO-4-(METHYL AMINO)BENZOYL}(PYRIDIN-2-YL)AMINO]-PROPANOATE 212322-56-0
4-CYNO PHENYL GLYCINE 42288-26-6
18 EFINACONAZOLE 4-METHYLIDENE PIPERIDINEHYDROCHLORIDE 144230-50-2
19 EDOXABAN 5-METHYL-4,5,6,7-TETRAHYDROTHIAZOLO[5,4-C]PYRIDINE-2-CARBOXYLIC ACID HCL 720720-96-7
2-AMINO-5-METHYL-4,5,6,7-TETRAHYDROTHIAZOLO[5,4-C]PYRIDINE 17899-48-8
5-METHYL-4,5,6,7-TETRAHYDROTHIAZOLE [5,4-C]PYRIDINE TOSYLATE 259809-24-0
2-BROMO-5-METHYL-4,5,6,7-TETRAHYDROTHIAZOLO[5,4-C]PYRIDINE TOSYLATE 143150-92-9
2-[(5-CHLOROPYRIDIN-2-YL)AMINO]-2-OXOACETIC ACID ETHYL ESTER HCI 1243308-37-3
20 ELTROMBOPAG 3,4-DIMETHYLPHENYLHYDRAZINE HCl 60481-51-8
(2-BROMO-6-NITROPHENOL) 13073-25-1
2-(3,4-DIMETHYLPHENYL)-5-METHYL-2,4-DIHYDRO-3H-PYRAZOL-3- ONE 277211-70-4
21 ERLOTINIB ETHYL-2-AMINO-4,5-BIS-(2-METHOXYETHOXY) BENZOATE HCl 183322-17-0
6,7-BIS-(2-METHOXYETHOXY)-4(3H)-QUINAZOLINONE 179688-29-0
22 FLIBANSERIN 1,3-DIHYDRO-2H-BENZIMIDAZOLE-2-ONE 615-16-7
1-ISOPROPENYL-2-BENZIMIDAZOLIDINONE 52099-72-6
1-(2-CHLOROETHYL)-1,3-DIHYDRO-2H-BENZIMIDAZOL-2-ONE 52548-84-2
1-(2-BROMOETHYL)-1,3-DIHYDRO-2H-BENZIMIDAZOL-2-ONE 103784-03-8
1-[3-(TRIFLUOROMETHYL)PHENYL]PIPERAZINE HCl 76835-14-8

4-[3-TRIFLUOROMETHYL)PHENYL]-1-(2-CHLOROETHYL) PIPERAZINE 57061-71-9 DIHYDROCHLORIDE

57061-71-9
23 FLORDIPINE 4-(2-AMINOETHYL)MORPHOLINE 42038-03-1
24 FORETINB CYCLOPROPANE-1 1-DICARBOXYLIC ACID 598-10-7
25 HYDRO CHLOROTHIAZIDE 5-CHLORO-2,4-DISULFAMOYLANILINE 121-30-2
26 LULICONAZOLE 1H-IMIDAZOL-1-YLACETONITRILE HYDROCHLORIDE 98873-55-3
1-(CYANO METHYL) IMIDAZOLE HYDROCHLORIDE] 220476-15-3
2-BROMO-1-(2,4-DICHLOROPHENYL)ETHANONE 2631-72-3
27 LUMATEPERONE 2-BROMOPHENYLHYDRAZINE HYDROCHLORIDE 50709-33-6
2-CHLORO-N-METHYLACETAMIDE 96-30-0
4-PIPERIDONE MONOHYDRATE HYDROCHLORIDE 40064-34-4
N,N-DIMETHYL ETHYLENE DIAMINE 110-70-3
28 LOMITAPIDE 4-(N-BOC-AMINO) PIPERIDINE 73874-95-0
4-AMINO-N-BENZYL PIPERIDINE 50541-93-0
29 LABETALOL 5-(N,N-DIBENZYLGLYCYL)SALICYLAMIDE 30566-92-8
5-BROMOACETYL-SALICYLAMIDE 73866-23-6
30 MACITENTAN DIMETHYL(4-BROMOPHENYL)MALONATE 14906-35-4
5-(4-BROMOPHENYL)PYRIMIDINE-4,6-DIOL 706811-25-8
5-(4-BROMOPHENYL)-4,6-DICHLOROPYRIMIDINE 146533-41-7
2-HYDROXYPYRIMIDINE HCl 38353-09-2
5-BROMO-2-HYDROXYPYRIMIDINE 38353-06-9
5-BROMO-2-CHLOROPYRIMIDINE 32779-36-5
31 METYROSINE 4-BROMOPHENETOLE 588-96-5
N-METHYL-2,4-DINITRO ANILINE 2044-88-4
32 NAFTOPIDILE & URAPIDIL 1-(2-METHOXY PHENYL)PIPERAZINE HCl 5464-78-8
33 NINTEDANIB TRI METHYL ORTHO BENZOATE 707-07-3
TRI ETHYL ORTHO BENZOATE 1663-61-2
METHYL-4-CHLORO-3-NITRO BENZOIC ACID 14719-83-6
N-METHYL-4-NITROANILINE 100-15-2
2-CHLORO-N-METHYL-N-(4-NITROPHENYL)ACETAMIDE 2653-16-9
N-METHYL-2-(4-METHYLPIPERAZIN-1-YL)-N-(4-NITROPHENYL) ACETAMIDE 1139453-98-7
N-METHYL-2-(4-METHYLPIPERAZIN-1-YL)-N-(4AMINOPHENYL) ACETAMIDE 262368-30-9
METHYL 1-ACETYL-2-OXOINDOLINE-6-CARBOXYLATE 676326-36-6
1,3-DIMETHYL 2-[4-(METHOXYCARBONYL)-2-NITROPHENYL]PROPANEDIOATE 1160293-27-5
6-METHOXYCARBONYL-2-OXINDOLE 14192-26-8
2-BROMO-N-METHYL-N-(4-NITROPHENYL)ACETAMIDE 23543-31-9
34 OLAPARIB CYCLOPROPYL CARBONYL PIPERAZINE 59878-57-8
35 ORMELOXIFENE 1-(2-HYDROXY ETHYL)PYRROLIDINE 2955-88-6
36 OSPEMIFENE 2-(4-BROMOPHENOXY)TATRAHYDROPYRAN 36603-49-3
BENZYL-2-BROMOETHYLETHER 1462-37-9
2-(2-BROMOETHOXY)TETRAHYDROPYRAN 17739-45-6
37 POSACONAZOLE 1-(4-HYDROXYPHENYL)PIPERAZINE 56621-48-8
1-(4-HYRDOXYPHENYL)-4-(4-AMINO PHENYL)PIPERAZINE 74853-08-0
38 POMALIDOMIDE 3-NITROPHTHALIC ANHYDRIDE 641-70-3
39 PRUCALOPRIDE 1-CHLOR-3-METHOXYPROPANE 36215-07-3
1-(3-METHOXYPROPYL)PIPERIDIN-4-ONE 16771-85-0
1-(3-METHOXYPROPYL)PIPERIDIN-4-AMINE 179474-79-4
4-(N-BOC AMINO) PIPERIDINE 73874-95-0
40 PIMAVANSERIN 4-ISOBUTOXY BENZYLAMINE HCL SALT 37806-44-3
4-ISOBUTOXY BENZYLAMINE ACETATE 955997-89-4
4-ISOBUTOXY BENZALDEHYDE 18962-07-7
41 PAZOPANIB 5-AMINO-2-METHYLBENZENESULFONAMIDE 6973-09-7
2,4-DICHLORO PYRIMIDINE 3934-20-1
42 QUETIAPINE 1-[2-(2-HYDROXY ETHOXY)ETHYL]PIPERAZINE 13349-82-1
43 RIVAROXABAN 2-[[(5S)-2-OXO-3-[4-(3-OXO-4-MORPHOLINYL)PHENYL]-5- OXAZOLIDINYL]METHYL]-1H-ISOINDOLE-1,3(2H)-DIONE 446292-08-6
4-(4-NITROPHENYL)MORPHOLIN-3-ONE 446292-04-2
4-(4-AMINOPHENYL)MORPHOLIN-3-ONE

438056-69-0

S-(2,3-EPOXYPROPYL)PHTHALAMIDE 161596-47-0
44 RIBOCICLIB,
PALBOCICLIB
5-BROMO -2-NITRO PYRIDINE 39856-50-3
5-BROMO-2-CHLORO-N-CYCLOPENTYLPYRIMIDIN-4-AMINE 733039-20-8
45 RIBOCICLIB, PALBOCICLIB 5-BROMO-2,4-DICHLOROPYRIMIDINE 36082-50-5
5-BROMOURACIL 51-20-7
1-BOC- 4-(6-NITRO-3-PYRIDYL)PIPERAZINE 571189-16-7
1-BOC- 4-(6-AMINO-3-PYRIDYL)PIPERAZINE 571188-59-5
46 RIMONABANT 1-AMINO PIPERIDINE 2213-43-6
2,4-DICHLORO PHENYL HYDRAZINE HCL 5446-18-4
47 ROFLUMILAST 2-AMINO-3,5-DICHLOROPYRIDINE 22889-78-7
48 SELEXIPAG 5,6-DIPHENYLPYRAZIN-2-OL 18591-57-6
5-CHLORO-2,3-DIPHENYLPYRAZINE 41270-66-0
4-(ISOPROPYL AMINO)BUTANOL 42042-71-7
5-BROMO-2,3-DIPHENYLPYRAZINE 243472-70-0
49 TIOTROPIUM BROMIDE METHYL-2,2-DITHIENYL GLYCOLATE 26447-85-8
50 VILAZODONE ETHYL-5-PIPRAZINYL BENZOFURAN-2-CARBOXYLATE HCL 765935-67-9
ETHYL-5-NITROBENZOFURAN-2-CARBOXYLATE 69604-00-8
ETHYL-5-AMINO BENZOFURAN-2-CARBOXYLATE 174775-48-5
5-AMINOBENZOFURAN-2-CARBOXYLIC ACID 42933-44-8
5-PIPERAZINEYL-BENZOFURAN-2CARBOXAMIDE 183288-46-2
N,N-BIS(2-CHLOROETHYL)-4-METHYLBENZENE SULFONAMIDE 42137-88-2
51 VORTIOXETINE 2,4-DIMETHYL THIOPHENOL 13616-82-5
N-BOC-PIPERAZINE 57260-71-6
52 VILDAGLIPTIN 3-HYDROXY-1-ADAMANTAN AMINE 26447-85-8
    L-PROLINAMIDE 7531-52-4
53 VELBANAZINE (N,N-DIMETHYL AMINO METHYL)-5-METHYL-2-HEXANONE OXALATE SALT 2102090-17-3
54 ZONISAMIDE/ WARFARIN 4-HYDROXY COUMARINE 1076-38-6
55 AMLODIPINE N-(2-HYDROXYETHYL)PHTHALIMIDE 3891-07-4
56 BETRIXABAN N-(5-CHLOROPYRIDIN-2-YL)-5-METHOXY-2-NITROBENZAMIDE 280773-16-2
2-AMINO-N-(5-CHLOROPYRIDIN-2-YL)-5-METHOXYBENZAMIDE 280773-17-3

N-(5-CHLOROPYRIDIN-2-YL)-2-[(4-CYANOBENZOYL)AMINO]-5-METHOXYBENZAMIDE

330942-01-3
57 BILASTINE 2-(PIPERIDIN-4-YL)-1H—BENZIMIDAZOLE 38385-95-4
1-(2-ETHOXYETHYL)-2-(PIPERIDIN-4-YL)-1H-BENZO[D]IMIDAZOLE (FREE BASE) 110963-63-8
58 OSIMERTINIB 3-(2-CHLOROPYRIMIDIN-4-YL)-1-METHYLINDOLE 1032452-86-0
N,N,N'-TRIMETHYL ETHYLENE DIAMINE 142-25-6
2,4-DICHLORO PYRIMIDINE 3934-20-1
59 PYRANTEL & OXANTEL 1,2-DIMETHYL-1,4,5,6-TETRAHYDROPYRIMIDINE 4271-96-9
60 VALBENAZINE 3, 4- DIHYDRO- 6, 7- DIMETHOXY-ISOQUINOLINE 3382-18-1
3,4-DIHYDRO—6,7-DIMETHOXY-ISOQUINOLINE HYDROCHLORIDE 20232-39-7
61 LETERMOVIR 1-(3-METHOXYPHENYL) PIPERAZINE 16015-71-7
62 MILCICLIB 1-(4-AMINOPHENYL)-4-METHYLPIPERAZINE 16153-81-4
ETHYL (HYDROXYIMINO)CYANOACETATE 3849-21-6
63 RILPIVIRINE 4-IODO-2,6-DIMETHYLANILINE 4102-53-8
64 REPAGLINIDE N-ACETYL-L-GLUTAMICACID 1188-37-0
65 RANOLAZINE GUAIACOL GLYCIDYL ETHER 2210-74-4
66 SATAVAPTAN 4-(2-CHLORO ETHL)MORPHOLINE 3240-94-6
67 SACUBITRIL ETHYL-2-(TRIPHENYLPHOSPHORANYLIEDINE)PROPANOATE 5717-37-3
68 SORAFENIB 4-(4-AMINOPHENOXY)-N-METHYLPYRIDINE-2-CARBOXAMIDE 284462-37-9
4-CHLORO-(2-PYRIDYL)-N-METHYL CARBOXAMIDE 220000-87-3
69 ZONISAMIDE 1,2-BENZISOXAZOLE-3-ACETIC ACID 37924-67-7
70 CERITINIB / BRIGATINIB 2,4,5-TRICHLOROPYRMIDINE 5750-76-5
71 SUVOREXANT N-BOC-ETHYLENE DIAMINE 57260-73-8
72 FEDRATINIB 1-(2-CHLOROETHYL)PYRROLIDINEHCL 7250-67-1
3-AMINO-N-(TERT-BUTYL)BENZENESULPHONAMIDE 608523-94-0
73 TRILACICLIB 5-(4-METHYLPIPERAZIN-1-YL)PYRIDIN-2-AMINE 571189-49-6
74 FAVIPIRAVIR 6-BROMO-3-HYDROXYPYRAZINE-2-CARBOXAMIDE 259793-88-9
75 FAVIPIRAVIR 2-AMINOMALONAMIDE 62009-47-6
2,4-DIAMINOPYRIMIDINE 156-81-0
76 LOSARTAN 2-BUTYL-4-CHLORO-5-FORMYLIMIDAZOLE 83857-96-9
77 MOLNUPIRAVIR {(3AR,4R,6R,6AR)-6-[(4Z)-4-(HYDROXYIMINO)-2-OXO-3,4-DIHYDROPYRIMIDIN1(2H)-YL]-2,2-DIMETHYLTETRAHYDRO-2H-FURO[3,4-D][1,3]DIOXOL-4-YL}METHYL2METHYLPROPANOATE 2346620-55-9
78 CABOZANTINIB 1-((4-FLUOROPHENYL)CARBAMOYL)CYCLOPROPANE CARBOXYLIC ACID 849217-48-7
79 VILOXAZINE 2-[(2-ETHOXYPHENOXY)METHYL]OXIRANE 5296-35-5
80   5-BROMO-2-NITROPYRIDINE 39856-50-3
81   2-ETHYL-4-FLUORO NITROBENZENE 1089279-29-7
82 UMIFENOVIR ETHYL 5-HYDROXY-1,2-DIMETHYL-1H-INDOLE-3-CARBOXYLATE 15574-49-9
83 CLOMIPERAMINE 3-CHLORO-5-ACETYLIMINODIBENZYL 25961-11-9
84
 
 
TRAZODONE
 
 
1-(3-CHLORO PHENYL) PIPERAZINE 6640-24-0
1-(3-CHLORO PHENYL)4-(3-CHLORO PROPYL)PIPERAZINE HCL 52605-52-4
2H-[1,2,4] TRIAZOLO [4,3-A] PYRIDIN-3-ONE 6969-71-7
85
ENTACAPONE 3,4-DI HYDROXY 5-NITRO BENZYL DEHYDE 116313-85-0

* PATENT INFRINGMENT IS RESPONSIBILITY OF THE BUYER